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Current Topics in Pharmacology   Volumes    Volume 3 
Abstract
β-chloroethylamines discriminate between two distinct subtypes of M3-cholinoceptors, α1-adrenoceptors and histamine H1-receptors
Issei Takayanagi, Katsuo Koike
Pages: 1 - 34
Number of pages: 34
Current Topics in Pharmacology
Volume 3 

Copyright © 1997 Research Trends. All rights reserved

ABSTRACT
 
Muscarinic M3-receptors, α1-adrenoceptors and histamine H1-receptors can be divided into two subtypes discriminated by the β-chloroethylamines propylbenzilylcholine mustard (PrBCM), chloroethylclonidine (CEC) and phenoxybenzamine (PBZ), only in the presence of GTP of GTPγS. The full agonists interact with both subtypes to induce responses. The partial agonists activate one of them to induce responses but behave as competitive antagonists when they interact with the other. Figures (Fig. 8 and 18) in the full paper show the modification of the classical drug receptor mechanisms.
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